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Methyltetrazine-PEG5-NHS ester
CAS No. 1802907-92-1
Methyltetrazine-PEG5-NHS ester( —— )
Catalog No. M33430 CAS No. 1802907-92-1
Methyltetrazine-PEG5-NHS ester is a PROTAC linker belonging to the group of PEGs and is used for the synthesis of PROTAC molecules.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 43 | In Stock |
|
| 10MG | 65 | In Stock |
|
| 25MG | 117 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameMethyltetrazine-PEG5-NHS ester
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NoteResearch use only, not for human use.
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Brief DescriptionMethyltetrazine-PEG5-NHS ester is a PROTAC linker belonging to the group of PEGs and is used for the synthesis of PROTAC molecules.
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DescriptionMethyltetrazine-PEG5-NHS ester is a PEG-based PROTAC linker that can be used in the synthesis of PROTACs.
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In VitroPROTACs contain two different ligands connected by a linker; one is a ligand for an E3 ubiquitin ligase and the other is for the target protein. PROTACs exploit the intracellular ubiquitin-proteasome system to selectively degrade target proteins.
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In Vivo——
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Synonyms——
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PathwayPROTACs
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TargetPROTAC
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RecptorPROTAC Linker
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Research Area——
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Indication——
Chemical Information
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CAS Number1802907-92-1
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Formula Weight533.53
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Molecular FormulaC24H31N5O9
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Purity>98% (HPLC)
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Solubility——
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SMILESO=C(ON1C(=O)CCC1=O)CCOCCOCCOCCOCCOC=2C=CC(=CC2)C3=NN=C(N=N3)C
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. An S, et al. Small-molecule PROTACs: An emerging and promising approach for the development of targeted therapy drugs. EBioMedicine. 2018 Oct;36:553-562?
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